I-Pharmacodynamics ceftiofur yiklasi ye-β -lactam yamachiza okulwa ne-antibacterial, kunye nesenzo se-bactericidal esibanzi, esisebenzayo ngokuchasene ne-gram-positive kunye ne-gram-negative bacteria (kuquka ibhaktheriya evelisa i-β - lactamase). Indlela yayo yokulwa ne-antibacterial kukuthintela ukwakhiwa kodonga lweseli yebhaktiriya kwaye ikhokelele ekufeni kweebhaktheriya. Iibhaktheriya ezibuthathaka kakhulu ziyi-pasteurella multiplex, i-pasteurella hemolyticus, i-actinobacillus pleuropneumoniae, i-salmonella, i-escherichia coli, i-streptococcus, i-staphylococcus, njl njl. Ezinye i-pseudomonas aeruginosa, i-enterococcus resistant. Umsebenzi we-antibacterial wale mveliso unamandla kune-ampicillin, kwaye umsebenzi ochasene ne-streptococcus unamandla kune-fluoroquinolones.
I-Pharmacokinetics ceftiofur ifunxwa ngokukhawuleza nangokubanzi ngeenaliti ze-intramuscular kunye ne-subcutaneous, kodwa ayikwazi ukuwela umqobo wegazi lobuchopho. Uxinaniso lweziyobisi luphezulu egazini kunye nezicubu, kwaye ugxininiso lwegazi olusebenzayo lugcinwa ixesha elide. I-metabolite esebenzayo ye-desfuroylceftiofur inokuveliswa emzimbeni, kwaye iphinde ifakwe kwi-metabolized ibe yimveliso engasebenziyo ekhutshwe kumchamo kunye nendle.
β -lactam antibiotics. Isetyenziselwa ikakhulu ukunyanga izifo zebhaktiriya zemfuyo kunye neenkukhu. Ezifana neehagu ibhaktiriya yokuphefumla intsholongwane kunye nenkukhu escherichia coli, usulelo lwe-salmonella.
I-Ceftiofur isetyenziswa. Isitofu se-Intramuscular: I-dose enye, i-1.1- 2.2mg nge-1kg ubunzima bomzimba weenkomo, i-3-5mg yeegusha neehagu, i-5mg yenkukhu kunye nedada, kanye ngosuku ngeentsuku ze-3.
Isitofu esingaphantsi kwesikhumba: amantshontsho anosuku olu-1, i-0.1mg ngentsiba nganye.
(1) Inokubangela ukuphazamiseka kwezityalo zesisu okanye ukusuleleka kabini.
(2) Kukho i-nephrotoxicity ethile.
(3) Intlungu engapheliyo yendawo ingenzeka.
(1)Sebenzisa ngoku.
(2)Umthamo kufuneka ulungelelaniswe kwizilwanyana ezinokusilela kwezintso.
(3)Abantu abanovelwano kakhulu kwi-beta-lactam antibiotics kufuneka bakuphephe ukudibana nale mveliso kwaye bakuphephe ukuvezwa kubantwana.